Silk Road forums
Market => Product offers => Topic started by: Chancery on September 19, 2011, 12:06 am
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Nucynta 50mg. It's a new drug. Limited quantities in bundles of 5, 10 and max 20 pills. Price point of of $7.50 each. Looking for feedback on interest and price. US only.
Tapentadol (trade name Nucynta, Palexia, In India - ZYNTAP) Tapentadol is a new molecular entity that is structurally similar to tramadol (Ultram). It has opioid and nonopioid acitivity in a single compound. It is is a centrally acting analgesic with a dual mode of action as an agonist at the μ-opioid receptor and as a norepinephrine reuptake inhibitor. Tapentadol is FDA approved for the treatment of moderate to severe acute pain. Due to the dual mechanism of action as an opioid agonist and norepinephrine reuptake inhibitor, there is potential for off label use in chronic pain.
While its analgesic actions have been compared to tramadol and oxycodone, its general potency is somewhere between tramadol and morphine in effectiveness. Because Tapentadol is a selective serotonin and norepinephrine reuptake inhibitor (SNRI) it has properties that are similar to duloxetine (Cymbalta).
Its dual mode of action provides analgesia at similar levels of more potent narcotic analgesics such as hydrocodone, oxycodone, and meperidine with a more tolerable side effect profile.